SCHEMBL21296774

SCHEMBL21296774

CC(=O)Oc1ccc(Nc2cccc(-c3ccnn3C(=O)OC(C)(C)C)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.46
GAA P10253 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HSP90AA1 P07900 1/20 0.46
POLB P06746 2/20 0.36
KDM4E B2RXH2 1/20 0.36
JAK2 O60674 6/20 0.36
JAK1 P23458 5/20 0.36
LMNA P02545 3/20 0.36
KMT2A Q03164 2/20 0.36
JAK3 P52333 1/20 0.36
CYP17A1 P05093 1/20 0.36
SCN4A P35499 1/20 0.35
SCN3A Q9NY46 1/20 0.35
EGFR P00533 1/20 0.35
ITK Q08881 1/20 0.35
PKM P14618 1/20 0.35
HTT P42858 1/20 0.35
RECQL P46063 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21296776 0.87 KMT2A (0.53) MAPTALDH1A1POLBKDM4ELMNA
SCHEMBL23610572 0.83 KMT2A (0.54) MAPTALDH1A1POLBKDM4ELMNA
SCHEMBL21296779 0.78 JAK2 (0.43) MAPTALDH1A1POLBKDM4EJAK2
SCHEMBL21296800 0.76 CNR1 (0.43) ALDH1A1CYP17A1SCN4ASCN3ASCN9A
SCHEMBL21296840 0.76 ACP1 (0.42) JAK2JAK3
SCHEMBL23610573 0.75 SCN3A (0.44) MAPTLMNAKMT2ACYP17A1SCN4A
SCHEMBL21296771 0.75 MAP2K4 (0.39) MAPTHSP90AA1SCN4ASCN3ASCN9A
SCHEMBL23610577 0.74 HSD17B1 (0.47) POLBKMT2ASCN4ASCN3ASCN9A
SCHEMBL9110223 0.72 CYP17A1 (0.52) ALDH1A1CYP17A1TDP1
SCHEMBL21296839 0.72 PDK1 (0.48) POLBJAK2JAK1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019165158-A1 IL-6 INHIBITORS AND METHODS OF TREATMENT UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2019-08-29 WO disclosed