SCHEMBL213116

SCHEMBL213116

CC(=O)N(NCc1ccccc1Cl)[C@@H](CCC(=O)OCc1ccccc1)COC(=O)Nc1cc2ccccc2cn1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 2/20 0.37
MAP4K1 Q92918 1/20 0.36
PTGER1 P34995 4/20 0.36
MAPKAPK2 P49137 2/20 0.34
TSHR P16473 1/20 0.34
FSHR P23945 1/20 0.34
CTSK P43235 1/20 0.34
MAPK1 P28482 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
NOTUM Q6P988 1/20 0.33
GCK P35557 1/20 0.32
F2 P00734 1/20 0.32
WNT1 P04628 1/20 0.32
DYRK1A Q13627 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL210443 0.92 MAP4K1 (0.37) MAP4K1PTGER1MAPKAPK2TSHRFSHR
SCHEMBL212116 0.92 CTSK (0.36) CTSKALDH1A1NOTUM
SCHEMBL212590 0.91 CTSK (0.36) PTGER1CTSKALDH1A1NOTUMGCK
SCHEMBL212341 0.88 CTSK (0.37) CCKBRCTSKALDH1A1NOTUMGCK
SCHEMBL213515 0.87 CTSK (0.36) PTGER1MAPKAPK2CTSKALDH1A1NOTUM
SCHEMBL211462 0.87 CTSK (0.36) CTSKALDH1A1NOTUM
SCHEMBL2723695 0.87 MAP4K1 (0.38) CCKBRMAP4K1PTGER1MAPKAPK2TSHR
SCHEMBL210644 0.86 NOTUM (0.36) CTSKALDH1A1NOTUMGCK
SCHEMBL4353508 0.85 CTSK (0.37) CTSKMAPK1ALDH1A1NOTUMDYRK1A
SCHEMBL210077 0.85 NOTUM (0.36) CTSKMAPK1ALDH1A1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US claimed
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US disclosed