SCHEMBL21341995

SCHEMBL21341995

COc1cc(F)c(C2CCCN(C(=O)OC(C)(C)C)C2)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.46
SCN9A Q15858 1/20 0.46
TRPV3 Q8NET8 1/20 0.45
ALDH1A1 P00352 3/20 0.45
GPR119 Q8TDV5 2/20 0.44
MMP1 P03956 1/20 0.44
MMP9 P14780 1/20 0.44
MMP13 P45452 1/20 0.44
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HTT P42858 1/20 0.43
USP30 Q70CQ3 1/20 0.42
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
HPGDS O60760 1/20 0.42
STS P08842 2/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15649592 0.84 PDE4B (0.54) PDE4BALDH1A1MMP1MMP9MMP13
SCHEMBL21342033 0.80 PDE4B (0.45) PDE4BALDH1A1GPR119MEN1KMT2A
SCHEMBL21342468 0.80 PDE4B (0.45) PDE4BALDH1A1GPR119MEN1KMT2A
SCHEMBL21359263 0.78 BCL9 (0.60) PDE4BALDH1A1MEN1KMT2AUSP30
SCHEMBL19405061 0.78 GPR119 (0.52) PDE4BTRPV3GPR119MAPTUSP30
SCHEMBL28297784 0.78 KDM4E (0.50) PDE4BTRPV3GPR119MAPTHPGDS
SCHEMBL28297774 0.78 KDM4E (0.50) PDE4BTRPV3GPR119MAPTHPGDS
SCHEMBL31383614 0.77 ALDH1A1 (0.47) PDE4BTRPV3ALDH1A1MMP1MMP9
SCHEMBL15307876 0.77 KDM2B (0.57) ALDH1A1MAPTMEN1KMT2ASTS
SCHEMBL28782629 0.77 PDE4B (0.54) PDE4BSCN9AALDH1A1MMP1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170904-A1 PIPERIDINES OR PIPERIDONES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-09-12 WO disclosed