SCHEMBL21342012

SCHEMBL21342012

COc1ccc(C2CCC(=O)NC2)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.49
FPR1 P21462 5/20 0.44
FPR2 P25090 4/20 0.44
DDB1 Q16531 5/20 0.41
CRBN Q96SW2 5/20 0.41
PDE4A P27815 3/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
HTR2C P28335 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19559399 0.86 MTNR1A (0.64) MTNR1AFPR1FPR2PDE4APDE4B
SCHEMBL18117787 0.86 MTNR1A (0.64) MTNR1AFPR1FPR2PDE4APDE4B
SCHEMBL21342022 0.82 FPR1 (0.42) MTNR1AFPR1FPR2
SCHEMBL20010674 0.81 CPS1 (0.40) FPR1FPR2PDE4APDE4BPDE4C
SCHEMBL19988384 0.78 MTNR1A (0.49) MTNR1AFPR1FPR2PDE4APDE4B
SCHEMBL10736004 0.75 MTNR1A (0.43) MTNR1ADDB1CRBN
SCHEMBL21341944 0.75 HTR2A (0.55) HTR2C
SCHEMBL1529068 0.74 HTR2C (0.58) FPR1FPR2HTR2C
SCHEMBL11295068 0.74 DDB1 (0.43) MTNR1ADDB1CRBNPDE4APDE4B
SCHEMBL21342014 0.74 FPR1 (0.53) MTNR1AFPR1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170904-A1 PIPERIDINES OR PIPERIDONES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-09-12 WO disclosed