SCHEMBL2134676

SCHEMBL2134676

NC(=O)C(c1cccc(Cl)c1)c1ccccn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
GRM4 Q14833 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
NPC1 O15118 1/20 0.42
PKM P14618 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TRPM8 Q7Z2W7 3/20 0.41
S1PR2 O95136 1/20 0.41
S1PR4 O95977 1/20 0.41
S1PR3 Q99500 1/20 0.41
DOT1L Q8TEK3 3/20 0.41
KDR P35968 1/20 0.40
ACP3 P15309 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7759530 0.83 ALDH1A1 (0.64) ALDH1A1CYP1A2RAB9ASMN1; SMN2S1PR2
SCHEMBL639563 0.83 ALDH1A1 (0.64) ALDH1A1CYP1A2RAB9ASMN1; SMN2S1PR2
SCHEMBL19555119 0.83 ALDH1A1 (0.50) ALDH1A1CYP1A2RAB9AS1PR2S1PR4
Hydrochloric Acid SCHEMBL4200885 0.82 ALDH1A1 (0.62) ALDH1A1CYP1A2RAB9ASMN1; SMN2S1PR2
Hydrochloric Acid SCHEMBL27529639 0.82 ALDH1A1 (0.62) ALDH1A1CYP1A2RAB9ASMN1; SMN2S1PR2
SCHEMBL6436240 0.80 CYP1A2 (0.43) ALDH1A1CYP1A2GRM4S1PR3SLC6A2
SCHEMBL29893620 0.79 AURKA (0.40)
SCHEMBL28889316 0.79 AURKA (0.40)
SCHEMBL23366716 0.77 SLC6A2 (0.46) GRM4HDAC6NFKB1S1PR2S1PR4
SCHEMBL132880 0.77 SLC6A2 (0.46) ALDH1A1CYP1A2GRM4HDAC6S1PR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9463187-B2 Methylphenidate derivatives and uses of them AMPIO PHARMACEUTICALS, INC. (US) 2016-10-11 US disclosed
US-20120101129-A1 Methylphenidate Derivatives and Uses of Them AMPIO PHARMACEUTICALS, INC. 2012-04-26 US disclosed
US-8076485-B2 Methylphenidate derivatives and uses of them INSTITUTE FOR MOLECULAR MEDICINE, INC. (US) 2011-12-13 US disclosed
US-7459467-B2 Manufacturing process for methyl phenidate and intermediates thereof IPCA LABORATORIES, LTD. (IN) 2008-12-02 US disclosed
EP-1607388-B1 An improved manufacturing process for methylphenidate and intermediates thereof IPCA LAB LTD (IN) 2008-02-20 EP disclosed
EP-1607388-A1 An improved manufacturing process for methylphenidate and intermediates thereof IPCA Laboratories Limited (IN) 2005-12-21 EP disclosed
US-20050277667-A1 Manufacturing process for methyl phenidate and intermediates thereof IPCA LABORATORIES LIMITED (IN) 2005-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050277667-A1 Manufacturing process for methyl phenidate and intermediates thereof COMT, ADH1C, CYP4B1 ALDH1A1 109/4885CYP1A2 20/4885GRM4 256/4885
US-20120101129-A1 Methylphenidate Derivatives and Uses of Them SLC6A3, COMT, UGT1A1 ALDH1A1 335/4885CYP1A2 22/4885GRM4 82/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.