SCHEMBL21358147

SCHEMBL21358147

CC1(C)OB(CCCC2CCN(C(=O)OCc3ccccc3)C2CO)OC1(C)C

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
F2 P00734 2/20 0.39
ELANE P08246 2/20 0.39
CTSG P08311 1/20 0.39
PREP P48147 2/20 0.39
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21367041 0.86 TP53 (0.40) SMN1; SMN2NPC1RAB9AF2ELANE
SCHEMBL22118726 0.86 TP53 (0.40) SMN1; SMN2NPC1RAB9AF2ELANE
SCHEMBL31367114 0.86 TP53 (0.40) SMN1; SMN2NPC1RAB9AF2ELANE
SCHEMBL21358644 0.78 MITF (0.36) SMN1; SMN2NPC1RAB9APREP
SCHEMBL16329051 0.78 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9AELANEPREP
SCHEMBL31367163 0.77 HTT (0.37) SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL21358090 0.76 PDE4B (0.46) SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL31367121 0.75 SMN1; SMN2 (0.40) SMN1; SMN2NPC1RAB9APREPCYP2C19
SCHEMBL21358094 0.75 PDK1 (0.36) SMN1; SMN2NPC1RAB9APREP
SCHEMBL31367151 0.74 HTR2C (0.43) SMN1; SMN2NPC1RAB9ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3765006-A1 ARGINASE INHIBITORS AND METHODS OF USE Merck Sharp&Dohme Corp. (US) 2021-01-20 EP disclosed
WO-2019177873-A1 ARGINASE INHIBITORS AND METHODS OF USE MERCK SHARP & DOHME CORP. (US) 2019-09-19 WO disclosed