SCHEMBL21362443

SCHEMBL21362443

COc1cc(C(=O)c2ccc(C[S+]([O-])N(C)C(=O)OC(C)(C)C)cc2Br)ccc1F

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 1/20 0.35
ACHE P22303 6/20 0.35
BCHE P06276 3/20 0.33
ALDH1A1 P00352 1/20 0.33
MTNR1A P48039 3/20 0.31
MTNR1B P49286 3/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158172 0.81 ALDH1A1 (0.39) TAS2R14ACHEALDH1A1ROCK2ROCK1
SCHEMBL20157608 0.76 ALDH1A1 (0.44) TAS2R14ACHEBCHEALDH1A1
SCHEMBL21362768 0.75 PPARG (0.36) ALDH1A1MTNR1AMTNR1BROCK2ROCK1
SCHEMBL21362766 0.72 ALDH1A1 (0.41) ACHEALDH1A1ROCK2ROCK1
SCHEMBL21351917 0.72 ALDH1A1 (0.40) TAS2R14ACHEALDH1A1MAPT
SCHEMBL20157679 0.72 ALDH1A1 (0.40) TAS2R14ACHEALDH1A1ROCK2ROCK1
SCHEMBL20157681 0.72 ALDH1A1 (0.40) ACHEALDH1A1ROCK2ROCK1MAPT
SCHEMBL20157726 0.71 ACHE (0.34) ACHEBCHEALDH1A1MTNR1AMTNR1B
SCHEMBL20157484 0.70 ALDH1A1 (0.48) ALDH1A1MAPT
SCHEMBL20158056 0.70 ACHE (0.35) ACHEBCHEALDH1A1MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed