SCHEMBL20158056

SCHEMBL20158056

CCc1ccc(C(=O)c2ccc(CS(=O)(=O)N(C)C(=O)OC(C)(C)C)cc2Br)cc1OC

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACHE P22303 8/20 0.35
BCHE P06276 5/20 0.35
MTNR1A P48039 2/20 0.34
MTNR1B P49286 2/20 0.34
ALDH1A1 P00352 1/20 0.33
HDAC8 Q9BY41 1/20 0.31
PDF Q9HBH1 1/20 0.31
HTT P42858 1/20 0.31
CYP1A2 P05177 3/20 0.31
CYP2C19 P33261 3/20 0.31
CYP3A4 P08684 2/20 0.31
TSHR P16473 2/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
KMT2A Q03164 1/20 0.31
AAK1 Q2M2I8 1/20 0.31
CYP2D6 P10635 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157726 0.90 ACHE (0.34) ACHEBCHEMTNR1AMTNR1BALDH1A1
SCHEMBL21362523 0.88 ACHE (0.33) ACHEBCHEMTNR1AMTNR1BALDH1A1
SCHEMBL20158055 0.83 CA12 (0.38) ACHEBCHEMTNR1AMTNR1BALDH1A1
SCHEMBL21564703 0.76 MAPT (0.33) ALDH1A1HTTMEN1LMNAKMT2A
SCHEMBL21550462 0.75 NPC1 (0.36) ALDH1A1MEN1LMNAKMT2AHPGD
SCHEMBL20158011 0.72 CA12 (0.38) ACHEBCHEMTNR1AMTNR1BALDH1A1
SCHEMBL20157485 0.71 ALDH1A1 (0.41) ACHEBCHEALDH1A1PDFCYP1A2
SCHEMBL21557859 0.70 ALDH1A1 (0.40) ACHEBCHEALDH1A1HDAC8PDF
SCHEMBL20157679 0.70 ALDH1A1 (0.40) ACHEALDH1A1PDFCYP1A2CYP2C19
SCHEMBL21362443 0.70 TAS2R14 (0.35) ACHEBCHEMTNR1AMTNR1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed