SCHEMBL21362597

SCHEMBL21362597

CCCCc1ccc(C(=O)c2ccc(C)cc2)c(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LPL P06858 6/20 0.43
LIPG Q9Y5X9 6/20 0.43
PLK1 P53350 8/20 0.39
CNR2 P34972 1/20 0.39
PLK3 Q9H4B4 2/20 0.39
SRD5A2 P31213 1/20 0.37
RARB P10826 1/20 0.36
PPARA Q07869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362596 0.90 LPL (0.42) LPLLIPGPLK1CNR2RARB
SCHEMBL20157811 0.83 SRD5A2 (0.36) SRD5A2
SCHEMBL20157690 0.82 SRD5A2 (0.37) SRD5A2
SCHEMBL20158134 0.81 SRD5A2 (0.35) SRD5A2
SCHEMBL20157897 0.80 SRD5A2 (0.36) SRD5A2
SCHEMBL21362721 0.79 SRD5A2 (0.35) SRD5A2
SCHEMBL5414465 0.78 LPL (0.55) LPLLIPGPLK1PLK3RARB
SCHEMBL20157444 0.77 MEN1 (0.37) LPLLIPGPLK1CNR2
SCHEMBL20157806 0.76 HTT (0.49)
SCHEMBL23510046 0.76 LIPG (0.49) LPLLIPGPLK1RARBPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed