SCHEMBL21362596

SCHEMBL21362596

CCCCc1ccc(C(=O)c2ccc(F)cc2)c(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LPL P06858 6/20 0.42
LIPG Q9Y5X9 6/20 0.42
CXCR2 P25025 4/20 0.39
PLK1 P53350 1/20 0.39
HTR7 P34969 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CNR2 P34972 1/20 0.36
AGTR1 P30556 2/20 0.36
AGTR2 P50052 2/20 0.36
RARB P10826 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362597 0.90 LPL (0.43) LPLLIPGPLK1CNR2RARB
SCHEMBL21362722 0.84 CXCR2 (0.36) LPLLIPGCXCR2ALDH1A1LMNA
SCHEMBL20157420 0.83 CXCR2 (0.36) LPLLIPGCXCR2ALDH1A1LMNA
SCHEMBL20157831 0.83 CXCR2 (0.40) LPLLIPGCXCR2ALDH1A1LMNA
SCHEMBL20157565 0.83 LMNA (0.43) LPLLIPGCXCR2LMNA
SCHEMBL20157558 0.82 CXCR2 (0.37) LPLLIPGCXCR2
SCHEMBL20157904 0.82 CXCR2 (0.35) LPLLIPGCXCR2ALDH1A1LMNA
SCHEMBL21362081 0.81 CXCR2 (0.38) LPLLIPGCXCR2
SCHEMBL20157880 0.81 CXCR2 (0.36) LPLLIPGCXCR2ALDH1A1LMNA
SCHEMBL21362027 0.80 CXCR2 (0.35) LPLLIPGCXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed