SCHEMBL21362715

SCHEMBL21362715

C=Cc1ccc(C(O)c2cc(OC)c(F)cc2Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.40
GAA P10253 1/20 0.37
TUBB1 Q9H4B7 7/20 0.35
TOP2A P11388 1/20 0.34
TOP2B Q02880 1/20 0.34
KDM1A O60341 2/20 0.34
BACE1 P56817 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362021 0.86 ACHE (0.38) GAATOP2ATOP2B
SCHEMBL20157890 0.82 OPRK1 (0.35) GAATUBB1TOP2ATOP2B
SCHEMBL20157860 0.74 PDE10A (0.38) GAATOP2ATOP2B
SCHEMBL24826176 0.74 MGAM (0.40) GAA
SCHEMBL20157891 0.73 KDM1A (0.43) TRPA1TUBB1KDM1A
SCHEMBL6742136 0.72 LMNA (0.44) TRPA1
SCHEMBL11863667 0.71 CNR2 (0.47) GAATOP2ATOP2B
SCHEMBL20157931 0.71 GAA (0.38) GAATOP2ATOP2B
SCHEMBL20157895 0.69 TOP2A (0.37) GAATOP2ATOP2B
SCHEMBL20157992 0.69 TOP2A (0.40) GAATUBB1TOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed