SCHEMBL20158058

SCHEMBL20158058

COc1cc(C(=O)c2ccc(CS(N)(=O)=O)cc2Br)ccc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
SLC22A6 Q4U2R8 1/20 0.39
SLC22A8 Q8TCC7 1/20 0.39
TSHR P16473 2/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 2/20 0.37
PKM P14618 2/20 0.37
CYP2D6 P10635 1/20 0.37
USP2 O75604 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
PDF Q9HBH1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157485 0.89 ALDH1A1 (0.41) ALDH1A1SLC22A6SLC22A8TSHRCYP1A2
SCHEMBL21351917 0.88 ALDH1A1 (0.40) ALDH1A1SLC22A6SLC22A8TSHRCYP1A2
SCHEMBL21362793 0.84 PKM (0.49) ALDH1A1SLC22A6SLC22A8TSHRCYP1A2
SCHEMBL20157609 0.84 ALDH1A1 (0.46) ALDH1A1SLC22A6SLC22A8TSHRCYP1A2
SCHEMBL20158011 0.81 CA12 (0.38) ALDH1A1CYP1A2CYP2C19MAPTGAA
SCHEMBL20157726 0.80 ACHE (0.34) ALDH1A1TSHRCYP1A2CYP2C19CYP3A4
SCHEMBL20157483 0.79 ALDH1A1 (0.50) ALDH1A1SLC22A6SLC22A8TSHRCYP1A2
SCHEMBL21351905 0.77 CA2 (0.41) TSHRMAPTCA1CA2CA7
SCHEMBL21557859 0.76 ALDH1A1 (0.40) ALDH1A1TSHRCYP1A2CYP2C19CYP3A4
SCHEMBL20157679 0.76 ALDH1A1 (0.40) ALDH1A1TSHRCYP1A2CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed