SCHEMBL21382863

SCHEMBL21382863

CCOc1ccn(-c2cccc(OC)c2)c(=O)c1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
TP53 P04637 2/20 0.47
GRM1 Q13255 1/20 0.45
KMT2A Q03164 2/20 0.43
MAPT P10636 2/20 0.43
ALKBH5 Q6P6C2 1/20 0.43
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
NOTUM Q6P988 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21385290 0.86 MEN1 (0.45) HPGDTP53GRM1KMT2AMAPT
SCHEMBL15506038 0.86 GLA (0.43) ALDH1A1KMT2ANOTUMLMNA
SCHEMBL21383448 0.86 AXL (0.43) ALDH1A1NOTUM
SCHEMBL16366161 0.79 LMNA (0.41) KDM4EALDH1A1TP53GRM1KMT2A
SCHEMBL22234532 0.78 MET (0.43) TP53RXFP1
SCHEMBL721541 0.78 MET (0.50) KDM4EALDH1A1HPGDTP53MAPT
SCHEMBL21383502 0.78 MET (0.43) KDM4EALDH1A1GRM1KMT2AMAPT
SCHEMBL15506073 0.76 CA12 (0.51) KDM4EALDH1A1HPGDKMT2AMAPT
SCHEMBL21385115 0.76 CYP1A2 (0.41)
SCHEMBL23749466 0.75 AXL (0.43) ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3762392-B1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO LTD (KR) 2024-05-15 EP disclosed
US-11447500-B2 Thienopyridine derivatives and pharmaceutical composition comprising same WELLMARKER BIO CO., LTD. (KR) 2022-09-20 US disclosed
US-20220288043-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO, LTD. (KR) 2022-09-15 US disclosed
CN-111295386-B Thienopyridine derivatives and pharmaceutical compositions containing the same 伟迈可生物有限公司 2022-09-06 CN disclosed
US-20210317133-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO., LTD. (KR) 2021-10-14 US disclosed
US-20210317133-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO., LTD. (KR) 2021-10-14 US disclosed
EP-3762392-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME Wellmarker Bio Co., Ltd. (KR) 2021-01-13 EP disclosed
CN-111295386-A Thienopyridine derivatives and pharmaceutical compositions containing the same 伟迈可生物有限公司 2020-06-16 CN disclosed
WO-2019182274-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO., LTD. (KR) 2019-09-26 WO disclosed
WO-2019182274-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME WELLMARKER BIO CO., LTD. (KR) 2019-09-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11447500-B2 Thienopyridine derivatives and pharmaceutical composition comprising same MAP4K5, MAP4K2, MAP3K9 KDM4E 2286/4885ALDH1A1 2254/4885HPGD 496/4885
US-20210317133-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME MAP4K5, MAP4K2, MAP3K9 KDM4E 2286/4885ALDH1A1 2254/4885HPGD 496/4885
US-20220288043-A1 THIENOPYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING SAME PRKACA, MAP4K5, MAPKAPK5 KDM4E 2594/4885ALDH1A1 2359/4885HPGD 658/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.