Piperazine

Piperazine

SCHEMBL2138391

C1CNCCN1.OP(O)O

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Piperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.60
MAPT P10636 1/20 0.60
PDE4A P27815 1/20 0.60
KDR P35968 1/20 0.60
CXCR4 P61073 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
CYP2C9 P11712 1/20 0.38
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piperazine SCHEMBL9441873 0.95 HIF1A (0.55) HIF1AMAPTPDE4AKDRCXCR4
Piperazine SCHEMBL6306849 0.82 HIF1A (0.50) HIF1AMAPTPDE4AKDRCXCR4
Pyrrolidine SCHEMBL28835057 0.82
Piperidine SCHEMBL8528732 0.79 ALDH1A1 (0.69) HIF1AMAPTPDE4AKDRCXCR4
Piperidine SCHEMBL27278836 0.79 ALDH1A1 (0.69) HIF1AMAPTPDE4AKDRCXCR4
SCHEMBL2373879 0.78 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4
SCHEMBL577429 0.78 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4
SCHEMBL22003 0.78 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4
SCHEMBL3999265 0.78 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4
SCHEMBL5033222 0.78 HIF1A (1.00) HIF1AMAPTPDE4AKDRCXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7235604-B2 Polyamide- and polyolefin-based fire-retarded compositions ATOFINA (FR) 2007-06-26 US claimed
EP-1375594-B1 Flame retardant compositions based on polyamide and polyolefine ARKEMA (FR) 2005-12-14 EP claimed
CN-1215123-C Polyamide and polyolefine refractory composition ATOFINA (FR) 2005-08-17 CN claimed
US-20040054054-A1 Polyamide-and polyolefin-based fire-retarded compositions ANTOFINA (FR) 2004-03-18 US claimed
CN-1468906-A Polyamide and polyolefine refractory composition ���з��ɹ�˾ 2004-01-21 CN claimed
CN-1100439-A Flame-retardant compositions for mixtures of thermoplastic resins containing a zeolite and mixtures of thermoplastic resins including the said compositions ATOCHEM ELF SA (FR) 1995-03-22 CN claimed
EP-0286478-B1 PHOSPHOROUS-ACID SALTS, THEIR COMMPOSITIONS AND THEIR USE AS FIRE-PROOFING AGENTS ELF ATOCHEM S.A. (FR) 1993-03-10 EP claimed
US-12018140-B2 Flexible fire-retardant thermoplastic compositions having high thermomechanical strength, in particular for electric cables SK GEO CENTRIC CO., LTD. (KR) 2024-06-25 US disclosed
CN-105593340-B Flexible flameproof thermoplastic composition with high thermomechanical strength, in particular for electric cables 阿肯马法国公司 2020-11-03 CN disclosed
US-20160185942-A1 FLEXIBLE FIRE-RETARDANT THERMOPLASTIC COMPOSITIONS HAVING HIGH THERMOMECHANICAL STRENGTH, IN PARTICULAR FOR ELECTRIC CABLES ARKEMA FRANCE (FR) 2016-06-30 US disclosed
CN-105593340-A Flexible flameproof thermoplastic composition with high thermomechanical strength, in particular for electric cables ARKEMA FRANCE 2016-05-18 CN disclosed
US-7897673-B2 Flexible high thermomechanical stress-resistant and fireproof halogen-free thermoplastic compositions ARKEMA FRANCE (FR) 2011-03-01 US disclosed
US-20090253836-A1 FLEXIBLE HIGH THERMOMECHANICAL STRESS-RESISTANT AND FIREPROOF HALOGEN-FREE THERMOPLASTIC COMPOSITIONS ARKEMA FRANCE (FR) 2009-10-08 US disclosed
US-7235604-B2 Polyamide- and polyolefin-based fire-retarded compositions ATOFINA (FR) 2007-06-26 US disclosed
CN-1215123-C Polyamide and polyolefine refractory composition ATOFINA (FR) 2005-08-17 CN disclosed
US-20040054054-A1 Polyamide-and polyolefin-based fire-retarded compositions ANTOFINA (FR) 2004-03-18 US disclosed
CN-1468906-A Polyamide and polyolefine refractory composition ���з��ɹ�˾ 2004-01-21 CN disclosed
CN-1100439-A Flame-retardant compositions for mixtures of thermoplastic resins containing a zeolite and mixtures of thermoplastic resins including the said compositions ATOCHEM ELF SA (FR) 1995-03-22 CN disclosed
CN-1100438-A Zeolite containing composition for fireproof of synthetic resin and synthetic resin containing same ATOCHEM ELF SA (FR) 1995-03-22 CN disclosed
US-4879327-A PLASTICS ATOCHEM (FR) 1989-11-07 US disclosed