SCHEMBL21384565

SCHEMBL21384565

Cc1cc(Cl)cc(Nc2cc(F)c(C(F)(F)F)cc2Cl)c1NS(=O)(=O)C1CC1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.36
CCR2 P41597 7/20 0.36
BRAF P15056 1/20 0.34
CNR1 P21554 3/20 0.34
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
EPHX2 P34913 1/20 0.32
MRGPRX1 Q96LB2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384586 0.90 CNR2 (0.37) CNR2CCR2BRAFCNR1CYP11B1
SCHEMBL21394400 0.83 MRGPRX1 (0.44) SCN5ASCN9AMRGPRX1
SCHEMBL21394421 0.75 MRGPRX1 (0.46) MRGPRX1
SCHEMBL21384571 0.71 MRGPRX1 (0.60) MRGPRX1
SCHEMBL21384560 0.66 MCL1 (0.46) CNR2CCR2CNR1MRGPRX1
SCHEMBL21384575 0.66 MCL1 (0.46) CNR2CCR2CNR1MRGPRX1
SCHEMBL392514 0.65 MAP2K1 (0.43) CNR2BRAFCNR1MRGPRX1
SCHEMBL21384613 0.65 MRGPRX1 (0.61) MRGPRX1
SCHEMBL393515 0.65 BRAF (0.40) CNR2CCR2BRAFCNR1EPHX2
SCHEMBL21384561 0.64 ACLY (0.48) SCN5ASCN9AMRGPRX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed