SCHEMBL21384571

SCHEMBL21384571

O=C(Nc1cc(F)c(C(F)(F)F)cc1Cl)c1cc(Cl)ccc1NS(=O)(=O)C1CC1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 11/20 0.60
TP53 P04637 3/20 0.48
TSPO P30536 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 2/20 0.44
RAB9A P51151 2/20 0.44
HRH1 P35367 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TMPRSS4 Q9NRS4 2/20 0.43
POLB P06746 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
SLC10A2 Q12908 1/20 0.42
SLC10A1 Q14973 1/20 0.42
SLC10A6 Q3KNW5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384613 0.93 MRGPRX1 (0.61) MRGPRX1TP53TSPOKDM4EMAPT
SCHEMBL21394421 0.88 MRGPRX1 (0.46) MRGPRX1TP53TSPOKDM4EMAPT
SCHEMBL21394400 0.85 MRGPRX1 (0.44) MRGPRX1TP53TSPOKDM4EMAPT
SCHEMBL21384576 0.84 MRGPRX1 (0.63) MRGPRX1TSPOKDM4EHRH1TMPRSS4
SCHEMBL21381353 0.83 MRGPRX1 (0.62) MRGPRX1TSPOKDM4EMAPTRAB9A
SCHEMBL21394560 0.80 MRGPRX1 (0.51) MRGPRX1TP53TSPOMAPTHRH1
SCHEMBL21394361 0.80 MRGPRX1 (0.58) MRGPRX1TSPOMAPTTMPRSS4
SCHEMBL21394415 0.78 MRGPRX1 (0.61) MRGPRX1TSPOHRH1TMPRSS4SLC10A6
SCHEMBL21394554 0.77 MRGPRX1 (0.49) MRGPRX1TP53TSPOMAPTRAB9A
SCHEMBL21394417 0.76 MRGPRX1 (0.53) MRGPRX1TSPOHRH1TMPRSS4SLC10A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed