SCHEMBL21394400

SCHEMBL21394400

Cc1cc(Cl)cc(C(=O)Nc2cc(F)c(C(F)(F)F)cc2Cl)c1NS(=O)(=O)C1CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 9/20 0.44
TP53 P04637 2/20 0.41
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SCN9A Q15858 3/20 0.38
SCN5A Q14524 1/20 0.38
BCL2 P10415 1/20 0.38
KDM4E B2RXH2 1/20 0.38
TSPO P30536 1/20 0.37
TMPRSS4 Q9NRS4 3/20 0.37
HRH1 P35367 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21394421 0.91 MRGPRX1 (0.46) MRGPRX1TP53MAPTRAB9ASMN1; SMN2
SCHEMBL21384571 0.85 MRGPRX1 (0.60) MRGPRX1TP53MAPTRAB9ASMN1; SMN2
SCHEMBL21384565 0.83 CNR2 (0.36) MRGPRX1SCN9ASCN5A
SCHEMBL21384613 0.78 MRGPRX1 (0.61) MRGPRX1TP53MAPTRAB9ASMN1; SMN2
SCHEMBL21384586 0.75 CNR2 (0.37) MRGPRX1
SCHEMBL21384561 0.73 ACLY (0.48) MRGPRX1TP53SCN9ASCN5AKDM4E
SCHEMBL21384579 0.71 MRGPRX1 (0.41) MRGPRX1MAPTSCN9ASCN5A
SCHEMBL21384576 0.69 MRGPRX1 (0.63) MRGPRX1KDM4ETSPOTMPRSS4HRH1
SCHEMBL21394560 0.69 MRGPRX1 (0.51) MRGPRX1TP53MAPTTSPOTMPRSS4
SCHEMBL21381353 0.69 MRGPRX1 (0.62) MRGPRX1MAPTRAB9ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179436-A1 ACID AMIDE COMPOUND AND USE THEREOF IN TREATMENT OF CANCERS 成都海创药业有限公司 2019-09-26 WO disclosed