SCHEMBL21386554

SCHEMBL21386554

Cc1ccc(-c2ccc(N=C=S)c(C)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
LMNA P02545 1/20 0.38
NAAA Q02083 1/20 0.34
CYP3A4 P08684 4/20 0.33
TDP1 Q9NUW8 3/20 0.33
ADRA2A P08913 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TSHR P16473 1/20 0.33
AR P10275 1/20 0.33
HPGD P15428 2/20 0.33
MCL1 Q07820 1/20 0.33
ABCB11 O95342 1/20 0.32
NR3C1 P04150 1/20 0.32
CYP1A2 P05177 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ALOX15 P16050 1/20 0.32
ADRA2C P18825 1/20 0.32
MAOA P21397 1/20 0.32
DRD1 P21728 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18269958 1.00 ALDH1A1 (0.38) ALDH1A1LMNANAAACYP3A4TDP1
SCHEMBL1993331 0.92 ALDH1A1 (0.41) ALDH1A1LMNACYP3A4TDP1ADRA2A
SCHEMBL29305748 0.92 GRM5 (0.35) ALDH1A1LMNANAAACYP1A2
SCHEMBL21386559 0.85 GRM5 (0.35) ALDH1A1LMNANAAACYP1A2
SCHEMBL945304 0.84 NPC1 (0.46) ALDH1A1LMNACYP3A4TDP1ADRA2A
SCHEMBL30421135 0.84 NPC1 (0.46) ALDH1A1LMNACYP3A4TDP1ADRA2A
SCHEMBL29305779 0.84 CYP3A4 (0.35) ALDH1A1LMNACYP3A4ADRA2ANPC1
SCHEMBL14207004 0.82 NAAA (0.36) ALDH1A1LMNANAAAARCYP1A2
SCHEMBL12011023 0.82 NAAA (0.36) ALDH1A1LMNANAAAARCYP1A2
SCHEMBL29305752 0.81 FFAR1 (0.32) ALDH1A1LMNACYP3A4ADRA2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240072425-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2024-02-29 US disclosed
US-11834599-B2 Aromatic isothiocyanates MERCK PATENT GMBH (DE) 2023-12-05 US disclosed
US-11739265-B2 Aromatic isothiocyanates MERCK PATENT GMBH (DE) 2023-08-29 US disclosed
EP-3739020-B1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2023-08-23 EP disclosed
US-20230025385-A1 FLUORINATED AROMATIC COMPOUNDS MERCK PATENT GMBH (DE) 2023-01-26 US disclosed
WO-2022128845-A1 HETEROAROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed
US-11306251-B2 Liquid-crystalline medium MERCK PATENT GMBH (DE) 2022-04-19 US disclosed
US-11268026-B2 Liquid-crystalline medium MERCK PATENT GMBH (DE) 2022-03-08 US disclosed
WO-2022043376-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-03-03 WO disclosed
WO-2021116080-A1 AROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2021-06-17 WO disclosed
EP-3739020-A1 LIQUID-CRYSTALLINE MEDIUM Merck Patent GmbH (DE) 2020-11-18 EP disclosed
US-20200347301-A1 Isothiocyanato-tolanes MERCK PATENT GMBH (DE) 2020-11-05 US disclosed
EP-3733816-A1 ISOTHIOCYANATO-TOLANES Merck Patent GmbH (DE) 2020-11-04 EP disclosed
EP-3543313-B1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2020-10-07 EP disclosed
EP-3543314-B1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2020-09-09 EP disclosed
US-20190352564-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2019-11-21 US disclosed
US-20190292458-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2019-09-26 US disclosed
US-20190292460-A1 LIQUID-CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2019-09-26 US disclosed
EP-3543314-A1 LIQUID-CRYSTALLINE MEDIUM Merck Patent GmbH (DE) 2019-09-25 EP disclosed
EP-3543313-A1 LIQUID-CRYSTALLINE MEDIUM Merck Patent GmbH (DE) 2019-09-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240072425-A1 AROMATIC ISOTHIOCYANATES TRPA1, TRPC1, CRY1 ALDH1A1 1864/4885LMNA 2735/4885NAAA 3756/4885
US-20230025385-A1 FLUORINATED AROMATIC COMPOUNDS TRPA1, FOXM1, AFF1 ALDH1A1 1136/4885LMNA 2980/4885NAAA 3881/4885
US-11739265-B2 Aromatic isothiocyanates TRPA1, CRY1, FOXM1 ALDH1A1 1554/4885LMNA 4099/4885NAAA 3694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.