SCHEMBL21391038

SCHEMBL21391038

CC(O)(CC(=O)CCCc1nc2ccc(C#N)cc2n1C(C)(C)C(F)(F)F)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACSS2 Q9NR19 6/20 0.43
CCR9 P51686 2/20 0.33
SLC22A12 Q96S37 1/20 0.33
ALB P02768 1/20 0.33
BRD4 O60885 1/20 0.32
TBXA2R P21731 1/20 0.31
TLR8 Q9NR97 1/20 0.31
TLR7 Q9NYK1 1/20 0.31
PDE10A Q9Y233 1/20 0.31
AGTR1 P30556 1/20 0.31
AGTR2 P50052 1/20 0.31
TNKS O95271 1/20 0.31
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
HDAC6 Q9UBN7 1/20 0.30
APEX1 P27695 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21391037 0.97 ACSS2 (0.42) ACSS2CCR9SLC22A12ALBBRD4
SCHEMBL23132027 0.86 ACSS2 (0.34) ACSS2CCR9TLR8TLR7PDK1
SCHEMBL20110978 0.80 ACSS2 (0.45) ACSS2CCR9SLC22A12ALBPDK1
SCHEMBL18791849 0.80 ACSS2 (0.45) ACSS2CCR9SLC22A12ALBPDK1
SCHEMBL18791850 0.80 ACSS2 (0.45) ACSS2CCR9SLC22A12ALBPDK1
SCHEMBL21391043 0.78 ACSS2 (0.41) ACSS2CCR9SLC22A12ALBBRD4
SCHEMBL21390993 0.77 HTT (0.31) ACSS2AGTR1AGTR2
SCHEMBL21391062 0.76 ACSS2 (0.33) ACSS2
SCHEMBL21391052 0.76 ACSS2 (0.36) ACSS2BRD4
SCHEMBL21390959 0.75 TRPV4 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed