SCHEMBL21393582

SCHEMBL21393582

Cn1c(N)nc2cnn(C)c2c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 3/20 0.43
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
TRPA1 O75762 2/20 0.38
PRMT5 O14744 1/20 0.38
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.35
HPGD P15428 2/20 0.33
HTT P42858 2/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
ATM Q13315 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21393588 0.83 ALDH1A1 (0.41) KDM4EALDH1A1ADORA3ADORA2AADORA2B
SCHEMBL21363587 0.80 ALDH1A1 (0.39) KDM4EALDH1A1ADORA3ADORA2AADORA2B
SCHEMBL22477705 0.80 ALDH1A1 (0.39) KDM4EALDH1A1ADORA3ADORA2AADORA2B
SCHEMBL22477732 0.78 ALDH1A1 (0.38) KDM4EALDH1A1ADORA3ADORA2AADORA2B
SCHEMBL25165851 0.73 KDM4E (0.41) KDM4EALDH1A1ADORA3ADORA2AADORA2B
SCHEMBL30814728 0.70 TLR8 (0.39) ALDH1A1ADORA3ADORA2AADORA2BADORA1
SCHEMBL26155930 0.70 QTRT1 (0.42) KDM4EALDH1A1GLAHSD17B10LMNA
SCHEMBL4402726 0.68 KMT2A (0.41) KDM4EALDH1A1PRMT5CYP1A2POLB
SCHEMBL18255988 0.68 GRM4 (0.46) KDM4EALDH1A1ADORA3ADORA2AADORA2B
SCHEMBL21363488 0.66 ALDH1A1 (0.41) ALDH1A1ADORA2AADORA1TRPA1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019182925-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2019-09-26 WO disclosed