SCHEMBL30814728

SCHEMBL30814728

Cn1ncc2nc(N)n(CCCCCBr)c2c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 6/20 0.39
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
CXCR4 P61073 1/20 0.36
TRPA1 O75762 1/20 0.36
AGTR1 P30556 1/20 0.34
AGTR2 P50052 1/20 0.34
DPP4 P27487 3/20 0.34
PNP P00491 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 2/20 0.32
USP2 O75604 1/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30814548 0.79 TLR8 (0.44) TLR8CXCR4AGTR1AGTR2PNP
SCHEMBL4932058 0.78 TLR8 (0.49) TLR8CXCR4TRPA1AGTR1AGTR2
SCHEMBL30814463 0.71 AGTR1 (0.35) AGTR1AGTR2ALDH1A1
SCHEMBL21393582 0.70 KDM4E (0.49) ADORA3ADORA2AADORA2BADORA1TRPA1
SCHEMBL21393588 0.68 ALDH1A1 (0.41) ADORA3ADORA2AADORA2BADORA1TRPA1
SCHEMBL21363587 0.66 ALDH1A1 (0.39) ADORA3ADORA2AADORA2BADORA1TRPA1
SCHEMBL22477705 0.66 ALDH1A1 (0.39) ADORA3ADORA2AADORA2BADORA1TRPA1
SCHEMBL30814682 0.66 CXCR4 (0.81) TLR8CXCR4POLBHTT
SCHEMBL13217347 0.66 LMNA (0.43) AGTR1AGTR2DPP4ALDH1A1HPGD
SCHEMBL22477732 0.64 ALDH1A1 (0.38) ADORA3ADORA2AADORA2BADORA1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024046221-A1 EGFR INHIBITORS AND USES THEREOF DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2024-03-07 WO disclosed