SCHEMBL21394613

SCHEMBL21394613

Cc1nccc(C(=O)Nc2ccc(Cc3cccc(Cl)c3)cn2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
MAPK1 P28482 1/20 0.43
CNR2 P34972 1/20 0.43
LMNA P02545 1/20 0.43
ANO1 Q5XXA6 1/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 2/20 0.41
F10 P00742 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GRM4 Q14833 1/20 0.40
HCRTR1 O43613 1/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
SORT1 Q99523 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29357133 1.00 ALDH1A1 (0.48) ALDH1A1MAPK1CNR2LMNAANO1
SCHEMBL21394865 0.88 NR3C2 (0.47) ALDH1A1ANO1NPC1RAB9ASMN1; SMN2
SCHEMBL29358065 0.88 NR3C2 (0.47) ALDH1A1ANO1NPC1RAB9ASMN1; SMN2
SCHEMBL22479673 0.86 NPC1 (0.47) ALDH1A1MAPK1NPC1RAB9ASMN1; SMN2
SCHEMBL21395082 0.86 NPC1 (0.43) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL21394918 0.83 GRM5 (0.43) NPC1RAB9ASMN1; SMN2MAPTHCRTR1
SCHEMBL21394920 0.82 ALDH1A1 (0.49) ALDH1A1LMNANPC1RAB9AMAPT
SCHEMBL21394767 0.81 ALDH1A1 (0.47) ALDH1A1LMNANPC1RAB9ASMN1; SMN2
SCHEMBL29358525 0.81 ALDH1A1 (0.47) ALDH1A1LMNANPC1RAB9ASMN1; SMN2
SCHEMBL21395200 0.81 GRM4 (0.43) NPC1RAB9AGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084800-A Compounds and uses thereof 詹森药业有限公司 2024-05-28 CN disclosed
CN-118084801-A Compounds and uses thereof 詹森药业有限公司 2024-05-28 CN disclosed
CN-112312913-B Compounds and uses thereof 詹森药业有限公司 2024-03-08 CN disclosed
CN-114174273-A Compounds and uses thereof 优曼尼蒂治疗公司 2022-03-11 CN disclosed
CN-112312913-A Compounds and uses thereof 优曼尼蒂治疗公司 2021-02-02 CN disclosed
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed