SCHEMBL21395082

SCHEMBL21395082

Cc1nccc(C(=O)Nc2ccc(Cc3ccc(F)c(F)c3)cn2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
GRM5 P41594 2/20 0.40
GRM4 Q14833 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
PPARG P37231 1/20 0.40
CD38 P28907 1/20 0.39
WNT3A P56704 2/20 0.39
TP53 P04637 2/20 0.38
HCRTR1 O43613 1/20 0.38
MAPT P10636 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SORT1 Q99523 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22479673 0.92 NPC1 (0.47) NPC1RAB9AGRM5GRM4SMN1; SMN2
SCHEMBL21395200 0.88 GRM4 (0.43) NPC1RAB9AGRM5GRM4WNT3A
SCHEMBL29353664 0.88 GRM4 (0.43) NPC1RAB9AGRM5GRM4WNT3A
SCHEMBL21394918 0.88 GRM5 (0.43) NPC1RAB9AGRM5SMN1; SMN2WNT3A
SCHEMBL29358065 0.87 NR3C2 (0.47) NPC1RAB9AGRM5SMN1; SMN2WNT3A
SCHEMBL21394865 0.87 NR3C2 (0.47) NPC1RAB9AGRM5SMN1; SMN2WNT3A
SCHEMBL21395075 0.86 GRM5 (0.43) NPC1RAB9AGRM5GRM4SMN1; SMN2
SCHEMBL21394613 0.86 ALDH1A1 (0.48) NPC1RAB9AGRM4SMN1; SMN2TP53
SCHEMBL29357133 0.86 ALDH1A1 (0.48) NPC1RAB9AGRM4SMN1; SMN2TP53
SCHEMBL29356981 0.81 GPR6 (0.41) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed