SCHEMBL21394697

SCHEMBL21394697

Cn1c(C(=O)Nc2ccc(Cc3cc(F)cc(F)c3)cn2)coc1=O

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.39
ABCB1 P08183 2/20 0.36
ABCC1 P33527 1/20 0.36
NPY5R Q15761 6/20 0.36
KDM4E B2RXH2 2/20 0.36
GCK P35557 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 1/20 0.35
DEGS1 O15121 1/20 0.34
MEN1 O00255 1/20 0.34
RECQL P46063 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
NTRK1 P04629 1/20 0.34
GRM5 P41594 1/20 0.34
CSF1R P07333 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21394704 0.89 CACNA1H (0.37) AHRKDM4ENPC1RAB9ADEGS1
SCHEMBL21394991 0.82 AHR (0.42) AHRABCB1ABCC1NPY5RKDM4E
SCHEMBL21394956 0.77 AHR (0.44) AHRABCB1ABCC1KDM4ENPC1
SCHEMBL21394572 0.76 TSHR (0.44) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL21394958 0.76 P2RX3 (0.42) AHRABCB1ABCC1KDM4EGCK
SCHEMBL29356925 0.76 GCK (0.44) ABCB1ABCC1KDM4EGCKNPC1
SCHEMBL21394784 0.76 GCK (0.44) ABCB1ABCC1KDM4EGCKNPC1
SCHEMBL21394747 0.76 AHR (0.38) AHRABCB1ABCC1KDM4EGCK
SCHEMBL29357109 0.76 TSHR (0.44) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL21394981 0.75 SMN1; SMN2 (0.53) ABCB1ABCC1KDM4EDEGS1NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed