SCHEMBL21394956

SCHEMBL21394956

Cn1nccc(C(=O)Nc2ccc(Cc3cc(F)cc(F)c3)cn2)c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.44
ABCB1 P08183 2/20 0.41
KIT P10721 2/20 0.40
BRAF P15056 2/20 0.40
MAPK1 P28482 2/20 0.40
AKT1 P31749 2/20 0.40
KDR P35968 2/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
FGFR3 P22607 4/20 0.38
CSF1R P07333 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
AXL P30530 1/20 0.36
TYRO3 Q06418 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21395014 0.91 AHR (0.44) AHRKITBRAFMAPK1AKT1
SCHEMBL21395013 0.90 NPC1 (0.44) AHRKITBRAFMAPK1AKT1
SCHEMBL21395129 0.78 GRM5 (0.40) AHRABCB1NPC1RAB9AKDM4E
SCHEMBL29357109 0.78 TSHR (0.44) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL21394572 0.78 TSHR (0.44) NPC1RAB9AKDM4EALDH1A1SMN1; SMN2
SCHEMBL21394981 0.78 SMN1; SMN2 (0.53) ABCB1CSF1RKDM4EALDH1A1SMN1; SMN2
SCHEMBL21394697 0.77 AHR (0.39) AHRABCB1NPC1RAB9ACSF1R
SCHEMBL21394930 0.77 GRM5 (0.40) ABCB1NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL21394784 0.76 GCK (0.44) ABCB1NPC1RAB9AKDM4EALDH1A1
SCHEMBL21394991 0.76 AHR (0.42) AHRABCB1NPC1RAB9ACSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed