SCHEMBL21394713

SCHEMBL21394713

O=C(Nc1ccc(Cc2ccc(F)c(F)c2)cn1)c1cnc(Cl)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
JUN P05412 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
BRD4 O60885 1/20 0.42
KCNQ3 O43525 1/20 0.42
KCNQ2 O43526 1/20 0.42
KCNE1 P15382 1/20 0.42
KCNQ1 P51787 1/20 0.42
PPARG P37231 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
TSHR P16473 1/20 0.41
BACE1 P56817 8/20 0.40
BACE2 Q9Y5Z0 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21395025 0.89 NPC1 (0.45) NPC1RAB9ASMN1; SMN2TDP1BRD4
SCHEMBL21394955 0.87 RAB9A (0.44) NPC1RAB9ASMN1; SMN2KCNQ3KCNQ2
SCHEMBL21394947 0.87 JUN (0.43) NPC1RAB9ASMN1; SMN2JUNNFKB1
SCHEMBL21395078 0.87 CHEK1 (0.48) NPC1RAB9ASMN1; SMN2KCNQ3KCNQ2
SCHEMBL21395032 0.86 SMN1; SMN2 (0.42) NPC1RAB9ASMN1; SMN2JUNNFKB1
SCHEMBL21395072 0.85 NPC1 (0.42) NPC1RAB9ASMN1; SMN2JUNNFKB1
SCHEMBL21394702 0.82 MAOB (0.44) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL21394758 0.81 NPC1 (0.53) NPC1RAB9ASMN1; SMN2ALDH1A1BACE1
SCHEMBL21395182 0.81 GSK3B (0.44) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL29357852 0.81 NPC1 (0.53) NPC1RAB9ASMN1; SMN2ALDH1A1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed