SCHEMBL21395037

SCHEMBL21395037

N#Cc1cc(C(=O)Nc2ccc(Cc3cc(F)cc(F)c3)cn2)cnn1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GCK P35557 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
F10 P00742 1/20 0.38
CYP3A4 P08684 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
DEGS1 O15121 2/20 0.37
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
CHEK1 O14757 2/20 0.36
RARG P13631 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21394396 0.85 KCNQ3 (0.47) GCKKDM4EALDH1A1DEGS1KCNQ3
SCHEMBL21395030 0.84 NPC1 (0.45) GCKKDM4EABCB1ABCC1NPC1
SCHEMBL21394698 0.81 GCK (0.41) GCKKDM4EABCB1ABCC1NPC1
SCHEMBL21394932 0.81 CHEK1 (0.42) CHEK1
SCHEMBL21394694 0.80 GCK (0.42) GCKKDM4EABCB1ABCC1NPC1
SCHEMBL21394726 0.80 RAB9A (0.42) GCKNPC1ALDH1A1PKMTSHR
SCHEMBL21394654 0.80 WNT3A (0.44) GCKKDM4EABCB1ABCC1NPC1
SCHEMBL21394952 0.80 KCNQ3 (0.44) GCKCYP3A4SIRT2DEGS1KCNQ3
SCHEMBL21395023 0.80 DEGS1 (0.40) CYP3A4SIRT2DEGS1
SCHEMBL21395009 0.78 PARP1 (0.53) KDM4EABCB1ABCC1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed