SCHEMBL21395030

SCHEMBL21395030

O=C(Nc1ccc(Cc2cc(F)cc(F)c2)cn1)c1cnnc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
PKM P14618 1/20 0.45
TSHR P16473 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
F10 P00742 7/20 0.41
KDM4E B2RXH2 1/20 0.40
ABCB1 P08183 1/20 0.40
ABCC1 P33527 1/20 0.40
GCK P35557 1/20 0.39
KLKB1 P03952 2/20 0.39
DEGS1 O15121 1/20 0.39
CYP3A4 P08684 2/20 0.39
GRM5 P41594 1/20 0.39
BRD4 O60885 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21395037 0.84 GCK (0.39) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21394727 0.83 KMT2A (0.50) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21394654 0.83 WNT3A (0.44) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21394643 0.81 KDM4E (0.44) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21394947 0.81 JUN (0.43) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21395009 0.80 PARP1 (0.53) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21394395 0.79 KDM4E (0.49) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21394726 0.79 RAB9A (0.42) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21394393 0.79 NPC1 (0.43) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL29359205 0.76 MLLT1 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed