SCHEMBL21397243

SCHEMBL21397243

N#Cc1ccc(OCc2ccccc2)nc1Cl

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.51
CNR1 P21554 2/20 0.46
GRM5 P41594 2/20 0.43
SQOR Q9Y6N5 1/20 0.42
XDH P47989 2/20 0.41
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
PGGT1B P53609 1/20 0.41
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24668349 0.83 PDE2A (0.46) MAOBCNR1
SCHEMBL20571893 0.78 MAOB (0.44) MAOBCNR1GRM5SQORGABRG2
SCHEMBL30529379 0.78 MAOB (0.44) MAOBCNR1GRM5SQORGABRG2
SCHEMBL3432981 0.78 L3MBTL1 (0.47) XDHGABRG2GABRB3GABRA5GABRA3
SCHEMBL24497447 0.76 PKM (0.45) GRM5
SCHEMBL24497448 0.76 PKM (0.42) MAOBGRM5GABRG2GABRB3GABRA5
SCHEMBL3803814 0.75 GAA (0.39) XDH
SCHEMBL11994824 0.75 XDH (0.40) XDH
SCHEMBL1008560 0.73 KCNH2 (0.52) MAOBGRM5
SCHEMBL2959124 0.73 GABRA5 (0.55) MAOBGRM5SQORGABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183367-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed