SCHEMBL21414101

SCHEMBL21414101

Cc1ccc(-c2ccc3c4ccc(-c5ccc(C)cc5)cc4n(-c4cc(C#N)cc(-n5c6cc(-c7ccc(C)cc7)ccc6c6ccc(-c7ccc(C)cc7)cc65)c4-c4cc(C#N)cc(C#N)c4)c3c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
CYP2A6 P11509 1/20 0.37
CHEK1 O14757 1/20 0.37
AR P10275 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
MAOA P21397 3/20 0.34
MAOB P27338 3/20 0.34
PGR P06401 1/20 0.32
GRIA2 P42262 1/20 0.32
GRIA4 P48058 1/20 0.32
GRM5 P41594 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21414100 0.94 PDE9A (0.39) ALDH1A1CYP2A6CHEK1ARMAPKAPK2
SCHEMBL21414253 0.92 GRM5 (0.37) ALDH1A1CYP2A6CHEK1PGRGRM5
SCHEMBL21414227 0.92 ALDH1A1 (0.39) ALDH1A1CYP2A6MAOAMAOBGRM5
SCHEMBL21414262 0.92 CHEK1 (0.38) ALDH1A1CYP2A6CHEK1MAPKAPK2PGR
SCHEMBL21414144 0.91 PGR (0.36) CHEK1PGR
SCHEMBL21546479 0.91 GRIA2 (0.39) ALDH1A1CHEK1ARPGRGRIA2
SCHEMBL19913283 0.90 CHEK1 (0.37) ALDH1A1CYP2A6CHEK1ARMAPKAPK2
SCHEMBL20617164 0.89 RXRA (0.43) ALDH1A1CYP2A6CHEK1ARMAPKAPK2
SCHEMBL21414242 0.89 PGR (0.38) CHEK1PGRGRIA2GRIA4
SCHEMBL21414138 0.89 MAPKAPK2 (0.38) ALDH1A1CYP2A6CHEK1ARMAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3385264-B1 ORGANIC MOLECULES, IN PARTICULAR FOR THE APPLICATION IN ORGANIC OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2019-10-02 EP disclosed