SCHEMBL21415751

SCHEMBL21415751

CCSc1ccc(C(C)CC#N)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 9/20 0.43
MAOA P21397 2/20 0.43
PTGS2 P35354 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
MAOB P27338 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
PBRM1 Q86U86 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11072633 0.84 ESR1 (0.42) SLC6A4MAOAPTGS2PBRM1ESR1
SCHEMBL7379356 0.83 ESR1 (0.33) MAOAMAOBPBRM1ESR1ESR2
SCHEMBL12303200 0.81 SLC6A4 (0.44) SLC6A4MAOA
SCHEMBL18602333 0.81 SLC6A4 (0.44) SLC6A4MAOA
SCHEMBL171729 0.80 PTGS2 (0.42) SLC6A4MAOAPTGS2HTR2AHTR2C
SCHEMBL1104208 0.79 SLC6A4 (0.50) SLC6A4MAOA
SCHEMBL12303213 0.76 MAPK1 (0.33)
SCHEMBL626140 0.75 ACHE (0.44) LMNAPBRM1ESR1ESR2
SCHEMBL13175896 0.74 SLC6A4 (0.53) SLC6A4MAOAPTGS2MAOBTAS1R3
SCHEMBL25343596 0.73 ADRB2 (0.45) LMNAPBRM1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3207043-B3 DIHYDROPYRROLOPYRIDINE INHIBITORS OF ROR-GAMMA VITAE PHARMACEUTICALS LLC (US) 2019-10-02 EP disclosed