SCHEMBL21443572

SCHEMBL21443572

CCCc1ccnc(Cc2ccccc2)c1

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SREBF2 Q12772 2/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
HTR2B P41595 1/20 0.40
NR3C2 P08235 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CYP19A1 P11511 1/20 0.38
LTA4H P09960 1/20 0.38
CALM1 P0DP23 1/20 0.38
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11629366 0.85 LNPEP (0.46) L3MBTL1CYP19A1TDP1
SCHEMBL487201 0.81 KDM4E (0.56) SREBF2KDM4ELMNACYP3A4TSHR
SCHEMBL18924413 0.79 MME (0.39) TSHRHTR2BNR3C2L3MBTL1ALDH1A1
SCHEMBL2619306 0.79 CYP1A2 (0.47) SREBF2KDM4ELMNACYP3A4TSHR
SCHEMBL18924479 0.79 ESR1 (0.43) TSHRHTR2BNR3C2L3MBTL1CALM1
SCHEMBL13562418 0.78 NOS2 (0.53) KDM4EHTR2BL3MBTL1CALM1ALDH1A1
SCHEMBL5115091 0.78 RECQL (0.50) TSHRHTR2BL3MBTL1CALM1ALDH1A1
SCHEMBL24923570 0.77 SREBF2 (0.44) SREBF2KDM4ELMNACYP3A4TSHR
SCHEMBL18937949 0.76 L3MBTL1 (0.61) KDM4ELMNATSHRL3MBTL1ALDH1A1
SCHEMBL21686484 0.76 KDM4E (0.41) SREBF2KDM4ELMNACYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3549934-A1 HETEROARYL COMPOUNDS AND USES THEREOF Celgene CAR LLC (BM) 2019-10-09 EP disclosed