SCHEMBL21450366

SCHEMBL21450366

CC(C)(C)OC(=O)Nc1ccc(N)s1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.42
CA2 P00918 1/20 0.42
GAA P10253 1/20 0.40
PKM P14618 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP17A1 P05093 2/20 0.40
LCK P06239 3/20 0.39
PSMB8 P28062 1/20 0.38
MAP4K4 O95819 1/20 0.38
ATR Q13535 1/20 0.37
MAPKAPK2 P49137 1/20 0.36
GLS O94925 1/20 0.36
RAB9A P51151 1/20 0.35
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14364099 0.82 GAA (0.45) GAAPKMALOX15HSD17B10RAB9A
SCHEMBL206754 0.81 NFKB1 (0.50) CA1CA2GAAPKMALOX15
SCHEMBL26991593 0.80 LCK (0.42) CA1CA2GAAPKMALOX15
SCHEMBL28834445 0.80 LCK (0.41) CA1CA2GAAPKMALOX15
SCHEMBL1504066 0.80 ATR (0.43) CA1CA2GAAPKMALOX15
SCHEMBL13983816 0.79 LMNA (0.46) CA1CA2GAAPKMALOX15
SCHEMBL380080 0.79 DAO (0.42) CA1CA2GAAPKMALOX15
SCHEMBL380561 0.78 L3MBTL1 (0.49) CA1CA2GAAPKMALOX15
SCHEMBL15674780 0.78 LMNA (0.42) CA1CA2GAAPKMALOX15
SCHEMBL28070546 0.78 CYP17A1 (0.41) CA1CA2GAAPKMALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019193540-A1 HETEROARYL DERIVATIVES OF FORMULA (I) AS ATF4 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-10-10 WO disclosed