SCHEMBL28070546

SCHEMBL28070546

CCc1ccc(NC(=O)OC(C)(C)C)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.41
PSMB8 P28062 1/20 0.39
GAA P10253 2/20 0.38
PKM P14618 1/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 1/20 0.38
LCK P06239 2/20 0.37
MAPK14 Q16539 1/20 0.37
GLS O94925 1/20 0.37
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
AKT1 P31749 2/20 0.36
KCNQ4 P56696 1/20 0.36
KCNQ5 Q9NR82 1/20 0.36
NPC1 O15118 2/20 0.35
ATR Q13535 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28090827 0.88 CYP17A1 (0.41) CYP17A1PSMB8GAAPKMALOX15
SCHEMBL21199756 0.84 GLS (0.40) CYP17A1PSMB8GLSNPC1RAB9A
SCHEMBL206754 0.79 NFKB1 (0.50) CYP17A1PSMB8GAAPKMALOX15
SCHEMBL15674780 0.78 LMNA (0.42) CYP17A1PSMB8GAAPKMALOX15
SCHEMBL10266596 0.78 KDM4A (0.44) GAACA1CA2GLSCA12
SCHEMBL28834445 0.78 LCK (0.41) CYP17A1PSMB8GAAPKMALOX15
SCHEMBL26991593 0.78 LCK (0.42) CYP17A1PSMB8GAAPKMALOX15
SCHEMBL21450366 0.78 CA1 (0.42) CYP17A1PSMB8GAAPKMALOX15
SCHEMBL1504066 0.78 ATR (0.43) CYP17A1PSMB8GAAPKMALOX15
SCHEMBL8704326 0.77 HDAC3 (0.50) ALOX15HSD17B10KCNQ4KCNQ5NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658653-A Furo- and thieno-pyridine carboxamide compounds useful as PIM kinase inhibitors 因赛特公司 2016-06-08 CN disclosed