SCHEMBL21452403

SCHEMBL21452403

COc1cccc(C2(Cl)C[C@@H](C)CCC2=O)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SIGMAR1 Q99720 2/20 0.41
DDB1 Q16531 2/20 0.41
CRBN Q96SW2 2/20 0.41
MAPT P10636 1/20 0.40
ADAM17 P78536 1/20 0.40
GRIN2B Q13224 2/20 0.40
CTSD P07339 1/20 0.40
CTSE P14091 1/20 0.40
BACE1 P56817 1/20 0.40
ALDH1A1 P00352 2/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
SLC6A4 P31645 1/20 0.39
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452162 0.85 TAS1R3 (0.38) KDM1A
SCHEMBL21452371 0.82 CCR2 (0.41) MEN1KMT2ADDB1CRBNMAPT
SCHEMBL23003321 0.78 DDB1 (0.38) DDB1CRBNGRIN2BBACE1SLC6A4
SCHEMBL21452493 0.77 GRIN1 (0.46) KDM1AMEN1KMT2ASIGMAR1GRIN2B
SCHEMBL11189378 0.76 MEN1 (0.43) KDM1AMEN1KMT2AMAPTADAM17
SCHEMBL21452404 0.74 MEN1 (0.42) KDM1AMEN1KMT2ASIGMAR1ADAM17
SCHEMBL11186880 0.74 MAPT (0.44) MEN1KMT2AMAPTADAM17GRIN2B
SCHEMBL21452127 0.74 CHRM2 (0.38) MEN1KMT2ASIGMAR1DDB1CRBN
SCHEMBL11543846 0.73 ALDH1A1 (0.41) KDM1AMEN1KMT2AMAPTADAM17
SCHEMBL28255039 0.72 KDM1A (0.47) KDM1AMEN1KMT2AADAM17ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed