SCHEMBL21452371

SCHEMBL21452371

Cc1cccc(C2(Cl)C[C@@H](C)CCC2=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.41
HTR2C P28335 2/20 0.37
HTR2A P28223 1/20 0.37
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
NPSR1 Q6W5P4 2/20 0.36
POLB P06746 2/20 0.36
HTT P42858 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CHRNA1 P02708 1/20 0.35
CHRNG P07510 1/20 0.35
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
SLC6A2 P23975 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452403 0.82 KDM1A (0.46) MEN1KMT2ADDB1CRBNALDH1A1
SCHEMBL23003321 0.81 DDB1 (0.38) SLC6A2LMNADDB1CRBNHSD11B1
SCHEMBL21452162 0.78 TAS1R3 (0.38) HSD11B1
SCHEMBL21452488 0.75 HDAC4 (0.49) MEN1KMT2ANPSR1POLBHTT
SCHEMBL21452568 0.73 PDE2A (0.40) CCR2
SCHEMBL21452373 0.71 CCR2 (0.38) CCR2MEN1KMT2ANPSR1HTT
SCHEMBL21452182 0.71 MAOA (0.41) MEN1KMT2ASLC6A3DDB1CRBN
SCHEMBL23001592 0.71 MAOA (0.41) MEN1KMT2ASLC6A3DDB1CRBN
SCHEMBL21452127 0.69 CHRM2 (0.38) MEN1KMT2APOLBDDB1CRBN
SCHEMBL25839802 0.67 ACHE (0.46) CCR2HTR2CHTR2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed