SCHEMBL21452740

SCHEMBL21452740

COC(=O)c1cc2c(Br)cc(OCCNC(=O)c3c(F)cc(OC)cc3Br)cc2s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.38
RECQL P46063 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
ALDH1A1 P00352 2/20 0.36
PTPN2 P17706 1/20 0.35
LMNA P02545 1/20 0.34
RPS6KB1 P23443 1/20 0.34
CSNK1D P48730 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34
NTRK2 Q16620 1/20 0.34
AURKB Q96GD4 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
MTNR1A P48039 2/20 0.33
MTNR1B P49286 2/20 0.33
GPR35 Q9HC97 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18490302 0.78 OPRD1 (0.44) NPC1RAB9AL3MBTL1ALDH1A1PTPN2
SCHEMBL18490289 0.70 TBXAS1 (0.41) ALDH1A1PTPN2LMNAMEN1KMT2A
SCHEMBL26622018 0.69 PTPN2 (0.47) NPC1RAB9AL3MBTL1ALDH1A1PTPN2
SCHEMBL31550045 0.68 PTPN2 (0.43) NPC1RAB9AL3MBTL1ALDH1A1PTPN2
SCHEMBL3484110 0.67 STING1 (0.42) ALDH1A1CSNK1DGSK3AGSK3BDYRK1A
SCHEMBL9431415 0.66 RPS6KB1 (0.44) NPC1RAB9AL3MBTL1ALDH1A1PTPN2
SCHEMBL829006 0.66 CSNK2A2 (0.46) NPC1RAB9AALDH1A1PTPN2RPS6KB1
SCHEMBL21406179 0.65 STING1 (0.49) NPC1RAB9A
SCHEMBL26108710 0.63 MTNR1A (0.53) L3MBTL1ALDH1A1LMNAMTNR1AMTNR1B
SCHEMBL8017091 0.62 CYP3A4 (0.55) RAB9AL3MBTL1ALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019195124-A1 BENZOTHIOPHENES AND RELATED COMPOUNDS AS STING AGONISTS MERCK SHARP & DOHME CORP. (US) 2019-10-10 WO disclosed