Phosphoric Acid

Phosphoric Acid

SCHEMBL214567

C=C(C)CCc1nc(N)c2[nH]cnc2n1.O=P(O)(O)O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Phosphoric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR known ✓ P35968 1/20 0.37
DPP4 known ✓ P27487 1/20 0.35
MGMT P16455 6/20 0.44
CDK1 P06493 5/20 0.44
CCNB1 P14635 5/20 0.44
CCNA2 P20248 5/20 0.44
CDK2 P24941 5/20 0.44
CCNA1 P78396 5/20 0.44
PDPK1 O15530 1/20 0.43
GDA Q9Y2T3 1/20 0.43
POLA1 P09884 1/20 0.39
AURKB Q96GD4 1/20 0.37
PI4KA P42356 2/20 0.35
PI4K2B Q8TCG2 2/20 0.35
PI4K2A Q9BTU6 2/20 0.35
PI4KB Q9UBF8 2/20 0.35
LMNA P02545 1/20 0.35
DRD3 P35462 1/20 0.35
XDH P47989 1/20 0.35
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29677204 0.94 CDK2 (0.49) MGMTCDK1CCNB1CCNA2CDK2
SCHEMBL136630 0.94 CDK2 (0.49) MGMTCDK1CCNB1CCNA2CDK2
SCHEMBL25228360 0.89 MGMT (0.43) MGMTCDK1CCNB1CCNA2CDK2
SCHEMBL717431 0.82 CA5A (0.39) MGMTCDK1CCNB1CCNA2CDK2
SCHEMBL1024249 0.81 ADORA1 (0.35) MGMTCDK1CCNB1CCNA2CDK2
SCHEMBL30416185 0.80 PDPK1 (0.49) MGMTCDK1CCNB1CCNA2CDK2
Ribose (Furanose) SCHEMBL17275115 0.80 MGMT (0.38) MGMTCDK1CCNB1CCNA2CDK2
SCHEMBL15167310 0.79 TRPM2 (0.41)
SCHEMBL9656473 0.78 PDPK1 (0.46) MGMTCDK1CCNB1CCNA2CDK2
SCHEMBL15166956 0.78 TRPM2 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10676752-B2 Methods controlling gene expression BASF PLANT SCIENCE COMPANY GMBH (DE) 2020-06-09 US disclosed
US-9708619-B2 Methods for controlling gene expression using ta-siRNA BASF PLANT SCIENCE GMBH (DE) 2017-07-18 US disclosed
US-20160152994-A1 METHODS CONTROLLING GENE EXPRESSION BASF PLANT SCIENCE GMBH (DE) 2016-06-02 US disclosed
EP-2980220-A1 IMPROVED METHODS CONTROLLING GENE EXPRESSION BASF Plant Science GmbH (DE) 2016-02-03 EP disclosed
US-20150368663-A1 METHOD FOR ISOLATION OF TRANSCRIPTION TERMINATION SEQUENCES BASF PLANT SCIENCE GMBH (DE) 2015-12-24 US disclosed
US-9133466-B2 Method for isolation of transcription termination sequences BASF PLANT SCIENCE GMBH (DE) 2015-09-15 US disclosed
US-9085774-B2 Methods controlling gene expression BASF PLANT SCIENCE GMBH (DE) 2015-07-21 US disclosed
US-20140237683-A1 EXPRESSION ENHANCING INTRON SEQUENCES BASF PLANT SCIENCE GMBH (DE) 2014-08-21 US disclosed
US-8759506-B2 Expression enhancing intron sequences BASF PLANT SCIENCE GMBH (DE) 2014-06-24 US disclosed
EP-1874936-B1 IMPROVED METHODS CONTROLLING GENE EXPRESSION BASF PLANT SCIENCE GMBH (DE) 2013-10-30 EP disclosed
EP-1781784-A2 METHOD FOR ISOLATION OF TRANSCRIPTION TERMINATION SEQUENCES BASF Plant Science GmbH (DE) 2007-05-09 EP disclosed
WO-2007039454-A1 METHODS FOR CONTROLLING GENE EXPRESSION USING TA-SIRAN BASF PLANT SCIENCE GMBH (DE) 2007-04-12 WO disclosed
EP-1723241-A1 TRANSGENIC EXPRESSION CONSTRUCTS FOR VEGETATIVE PLANT TISSUE SPECIFIC EXPRESSION OF NUCLEIC ACIDS BASF Plant Science GmbH (DE) 2006-11-22 EP disclosed
WO-2006111512-A1 IMPROVED METHODS CONTROLLING GENE EXPRESSION BASF PLANT SCIENCE GMBH (DE) 2006-10-26 WO disclosed
WO-2006094976-A2 EXPRESSION ENHANCING INTRON SEQUENCES BASF PLANT SCIENCE GMBH (DE) 2006-09-14 WO disclosed
EP-1629096-A1 METHODS FOR ASSEMBLING MULTIPLE EXPRESSION CONSTRUCTS BASF Plant Science GmbH (DE) 2006-03-01 EP disclosed
WO-2006013072-A2 METHOD FOR ISOLATION OF TRANSCRIPTION TERMINATION SEQUENCES BASF PLANT SCIENCE GMBH (DE) 2006-02-09 WO disclosed
WO-2005108568-A1 METHODS FOR ASSEMBLING MULTIPLE EXPRESSION CONSTRUCTS BASF PLANT SCIENCE GMBH (DE) 2005-11-17 WO disclosed
WO-2005085450-A1 TRANSGENIC EXPRESSION CONSTRUCTS FOR VEGETATIVE PLANT TISSUE SPECIFIC EXPRESSION OF NUCLEIC ACIDS BASF PLANT SCIENCE GMBH (DE) 2005-09-15 WO disclosed
WO-2002034924-A2 EXPRESSION CASSETTE USED FOR THE TRANSGENIC EXPRESSION OF NUCLEIC ACIDS IN THE EMBRYONIC EPIDERMIS AND/OR FLOWER OF PLANTS BASF PLANT SCIENCE GMBH (DE) 2002-05-02 WO disclosed