SCHEMBL21470185

SCHEMBL21470185

C/C(C=O)=C\c1ccc(C(F)(F)F)nc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.44
TRPV4 Q9HBA0 1/20 0.42
TRPV1 Q8NER1 1/20 0.39
MAP4K4 O95819 1/20 0.35
PIK3CA P42336 1/20 0.35
KCNH2 Q12809 1/20 0.35
MINK1 Q8N4C8 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
PDE10A Q9Y233 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
TRPV3 Q8NET8 7/20 0.34
DAO P14920 1/20 0.33
DGAT1 O75907 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3469578 0.79 AKR1C3 (0.47) TRPV4TRPV1MRGPRX4DGAT1
SCHEMBL3469572 0.79 AKR1C3 (0.47) TRPV4TRPV1MRGPRX4DGAT1
SCHEMBL2401676 0.77 TRPV1 (0.50) TRPV4TRPV1
SCHEMBL2401668 0.77 TRPV1 (0.50) TRPV4TRPV1
SCHEMBL29417132 0.77 TRPV4 (0.52) ALDH1A1TRPV4TRPV1MAP4K4PIK3CA
SCHEMBL336320 0.77 TRPV4 (0.52) ALDH1A1TRPV4TRPV1MAP4K4PIK3CA
SCHEMBL7804952 0.74 ALDH1A1 (0.57) ALDH1A1TSHR
SCHEMBL3113876 0.74 TBXAS1 (0.47) TRPV4TRPV1MRGPRX4DGAT1
SCHEMBL3113886 0.74 TBXAS1 (0.47) TRPV4TRPV1MRGPRX4DGAT1
SCHEMBL30469174 0.74 MEN1 (0.43) ALDH1A1TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196714-A1 N-SUBSTITUTED ACRYLAMIDE DERIVATIVE AS DHODH INHIBITOR, AND PREPARATION AND USE THEREOF 华东理工大学 2019-10-17 WO disclosed