SCHEMBL21473716

SCHEMBL21473716

COC(=O)[C@@H](N)Cc1c(C)cc(C#N)cc1C

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 2/20 0.38
ALDH1A1 P00352 1/20 0.37
NLRP3 Q96P20 2/20 0.36
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
OPRK1 P41145 2/20 0.35
ANPEP P15144 1/20 0.35
CACNA1F O60840 1/20 0.34
CACNA1D Q01668 1/20 0.34
CACNA1S Q13698 1/20 0.34
CACNA1C Q13936 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL20236002 0.81 ALDH1A1 (0.43) ALDH1A1OPRM1
SCHEMBL5115246 0.81 OPRD1 (0.46) OPRM1OPRD1OPRK1
SCHEMBL5115242 0.81 OPRD1 (0.46) OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL20236003 0.81 ALDH1A1 (0.43) ALDH1A1OPRM1
Hydrochloric Acid SCHEMBL5775220 0.80 OPRD1 (0.46) OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL5775227 0.80 OPRD1 (0.46) OPRM1OPRD1OPRK1
SCHEMBL15705239 0.77 NLRP3 (0.38) GPR35NLRP3ANPEP
SCHEMBL24012345 0.77 ALDH1A1 (0.40) ALDH1A1OPRM1OPRD1OPRK1
SCHEMBL5569674 0.76 DPP4 (0.48) ALDH1A1NLRP3ANPEP
SCHEMBL16060347 0.76 DPP4 (0.48) ALDH1A1NLRP3ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019197274-A1 PROCESS FOR THE PREPARATION OF OPIOID MODULATORS QUIMICA SINTETICA, S. A. (ES) 2019-10-17 WO disclosed