SCHEMBL5115246

SCHEMBL5115246

COC(=O)C(N)Cc1c(C)cc(O)cc1C

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 9/20 0.46
OPRM1 P35372 7/20 0.46
OPRK1 P41145 6/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5115242 1.00 OPRD1 (0.46) OPRD1OPRM1OPRK1
Hydrochloric Acid SCHEMBL5775220 0.98 OPRD1 (0.46) OPRD1OPRM1OPRK1
Hydrochloric Acid SCHEMBL5775227 0.98 OPRD1 (0.46) OPRD1OPRM1OPRK1
SCHEMBL30162392 0.87 CYP3A4 (0.46) OPRD1OPRM1OPRK1
Hydrochloric Acid SCHEMBL20236002 0.87 ALDH1A1 (0.43) OPRM1
Hydrochloric Acid SCHEMBL20236003 0.87 ALDH1A1 (0.43) OPRM1
SCHEMBL25469337 0.85 OPRD1 (0.45) OPRD1OPRM1OPRK1
SCHEMBL21096380 0.83 OPRM1 (0.47) OPRD1OPRM1OPRK1
SCHEMBL21473716 0.81 GPR35 (0.38) OPRD1OPRM1OPRK1
SCHEMBL24012345 0.81 ALDH1A1 (0.40) OPRD1OPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439258-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM (CANADA) LTD (CA) 2008-10-21 US disclosed
US-7439258-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM (CANADA) LTD (CA) 2008-10-21 US disclosed
US-7439258-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM (CANADA) LTD (CA) 2008-10-21 US disclosed