SCHEMBL21481725

SCHEMBL21481725

Nc1nc(Cl)nc2c1cnn2Br

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
CDK1 P06493 1/20 0.39
PDE2A O00408 2/20 0.37
NT5E P21589 2/20 0.36
PI4KA P42356 1/20 0.33
PI4K2B Q8TCG2 1/20 0.33
PI4K2A Q9BTU6 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
KMT2A Q03164 1/20 0.31
CSNK1A1 P48729 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
GAA P10253 1/20 0.31
CFTR P13569 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29685062 0.78 PDE2A (0.60) CDK1PDE2API4KAPI4K2BPI4K2A
SCHEMBL130521 0.78 PDE2A (0.60) CDK1PDE2API4KAPI4K2BPI4K2A
SCHEMBL24500179 0.74 KDM4E (0.41) CDK1PDE2ANT5EPI4KAPI4K2B
SCHEMBL21481726 0.71 CDK1 (0.34) HTTCDK1PDE2ANT5E
SCHEMBL23274461 0.71 ALDH1A1 (0.59) PI4KAPI4K2BPI4K2API4KBKMT2A
SCHEMBL21481606 0.69 ADORA2A (0.52) HTTGAA
SCHEMBL31385338 0.69 ADORA2A (0.52) HTTGAA
SCHEMBL21481670 0.68 KDM4E (0.46)
SCHEMBL21481598 0.68 ADORA2A (0.39) HTTNT5E
SCHEMBL21462235 0.65 CYP3A4 (0.64) HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111433205-A Polycyclic compounds as allosteric SHP2 inhibitors 锐新医药公司 2020-07-17 CN disclosed
WO-2019196918-A1 FIVE-MEMBERED HETEROCYCLO-PYRIMIDINE COMPOUND, PHARMACEUTICAL COMPOSITION AND USE THEREOF 罗欣药业(上海)有限公司 2019-10-17 WO disclosed