SCHEMBL21495037

SCHEMBL21495037

C[Si](C)(C)C#Cc1ccc([C@H](Br)C=O)cc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1306384 0.74 GABRA1 (0.38) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8129656 0.74 ACACB (0.39) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1306505 0.72 APP (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL13397172 0.72 NR1H2 (0.31)
SCHEMBL17464776 0.72 ACACB (0.41)
SCHEMBL701214 0.72 CYP2A6 (0.43) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1535167 0.72 GSK3B (0.46)
SCHEMBL17464783 0.72 ACACB (0.41)
SCHEMBL3148515 0.71 ACACB (0.38) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL23977506 0.71 NOS3 (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019201865-A1 SUBSTITUTED AMINOTHIAZOLES AS INHIBITORS OF NUCLEASES MASARYKOVA UNIVERZITA (CZ) 2019-10-24 WO disclosed