SCHEMBL21496829

SCHEMBL21496829

COC(=O)C1(C)NCc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HTT P42858 1/20 0.40
ALDH1A1 P00352 4/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
POLB P06746 2/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28037815 0.84 ALDH1A1 (0.42) MEN1KMT2AALDH1A1CYP3A4POLB
SCHEMBL23183322 0.83 EPHX2 (0.39) MEN1KMT2ACYP3A4CYP2C19LMNA
SCHEMBL17648648 0.83 EPHX2 (0.39) MEN1KMT2ACYP3A4CYP2C19LMNA
SCHEMBL3696570 0.81 ALDH1A1 (0.44) ALDH1A1CYP3A4LMNAMAPTKDM4E
SCHEMBL3368929 0.78 ALDH1A1 (0.57) MEN1KMT2AHTTALDH1A1POLB
SCHEMBL547428 0.71 MEN1 (0.44) MEN1KMT2AHTTALDH1A1POLB
Bromide SCHEMBL10516381 0.70 MTNR1A (0.36) ALDH1A1CYP1A2LMNA
SCHEMBL15084239 0.70 ALDH1A1 (0.41) MEN1KMT2AALDH1A1CYP3A4CYP2C19
SCHEMBL3542185 0.69 ALDH1A1 (0.43) MEN1KMT2AALDH1A1CYP3A4CYP2C19
SCHEMBL1471124 0.69 PIN1 (0.53) MEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3784654-A1 ISOINDOLINES AS HDAC INHIBITORS Valo Early Discovery, Inc. (US) 2021-03-03 EP disclosed
WO-2019204550-A1 ISOINDOLINES AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2019-10-24 WO disclosed