SCHEMBL21508697

SCHEMBL21508697

O=c1[nH]c2ccncc2c(OCc2ccccc2)c1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.50
PARP1 P09874 3/20 0.49
CHEK1 O14757 2/20 0.48
HSD17B10 Q99714 2/20 0.45
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ACHE P22303 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14970200 0.84 HDAC1 (0.51) PARP1HSD17B10HDAC1HDAC6GABRP
SCHEMBL14968197 0.79 KDM4C (0.57) KDM4CPARP1CHEK1HSD17B10ALDH1A1
SCHEMBL14979958 0.79 PARP1 (0.43) KDM4CPARP1HSD17B10ACHEGRIN2D
SCHEMBL16106862 0.75 LMNA (0.45) PARP1HSD17B10HDAC1HDAC6ALDH1A1
SCHEMBL16107102 0.75 CTSV (0.44) HSD17B10ALDH1A1USP2TSHRCTSV
SCHEMBL14979997 0.72 CNR1 (0.50) HSD17B10HDAC1HDAC6ALDH1A1CTSV
SCHEMBL14969193 0.72 TMEM97 (0.44) HSD17B10HDAC1HDAC6CTSVCTSL
SCHEMBL14969243 0.72 KIF11 (0.44) HSD17B10HDAC1HDAC6ACHEALDH1A1
SCHEMBL14969170 0.71 ALDH1A1 (0.43) HSD17B10HDAC1HDAC6ALDH1A1USP2
SCHEMBL16107056 0.69 ALDH1A1 (0.50) HSD17B10ALDH1A1USP2TSHRCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2780026-B1 HCV NS3 PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2019-10-23 EP disclosed