SCHEMBL21550122

SCHEMBL21550122

CCS(=O)(=O)c1ccc(C(O)c2ccc(F)cc2Cl)c(Br)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
EPAS1 Q99814 3/20 0.38
MDM4 O15151 3/20 0.37
MDM2 Q00987 3/20 0.37
PSEN1 P49768 6/20 0.37
PSEN2 P49810 6/20 0.37
APH1B Q8WW43 6/20 0.37
NCSTN Q92542 6/20 0.37
APH1A Q96BI3 6/20 0.37
PSENEN Q9NZ42 6/20 0.37
APLNR P35414 1/20 0.36
RORC P51449 1/20 0.35
PKM P14618 1/20 0.34
POLB P06746 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.33
FDFT1 P37268 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21550133 0.86 ALDH1A1 (0.43) ALDH1A1PSEN1PSEN2APH1BNCSTN
SCHEMBL20157925 0.77 ALDH1A1 (0.36) ALDH1A1MDM2APLNRPKM
SCHEMBL21564721 0.77 MDM2 (0.30) MDM2
SCHEMBL21550148 0.76 PYGL (0.41) ALDH1A1EPAS1RORCPKMPOLB
SCHEMBL21550119 0.75 APLNR (0.35) MDM2APLNRPKMFDFT1
SCHEMBL21564723 0.74 MDM2 (0.31) MDM2
SCHEMBL28473298 0.74 MDM2 (0.46) MDM4MDM2
SCHEMBL21550018 0.72 MDM2 (0.49) ALDH1A1MDM4MDM2
SCHEMBL21550145 0.72 MDM2 (0.33) ALDH1A1MDM2PSEN1PSEN2APH1B
SCHEMBL28476113 0.70 MDM2 (0.39) MDM4MDM2APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed