SCHEMBL21551953

SCHEMBL21551953

CN(C)CCNC(=O)c1ccc(/C=C/c2ccc(Br)cc2Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
ALDH1A1 P00352 4/20 0.46
HPGD P15428 4/20 0.46
KDM4E B2RXH2 2/20 0.46
LMNA P02545 2/20 0.46
KDM1A O60341 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SETD7 Q8WTS6 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 1/20 0.44
ALOX12 P18054 1/20 0.44
ALOX5 P09917 1/20 0.43
HTT P42858 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
TP53 P04637 1/20 0.41
KMT2A Q03164 1/20 0.40
FLT3 P36888 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21551943 0.84 ALDH1A1 (0.51) CYP1A2ALDH1A1HPGDKDM4ELMNA
SCHEMBL1241975 0.79 ALDH1A1 (0.63) CYP1A2ALDH1A1HPGDKDM4ELMNA
SCHEMBL21551941 0.79 HDAC6 (0.62) MAPT
SCHEMBL21551949 0.79 SMN1; SMN2 (0.58) CYP1A2ALDH1A1HPGDSMN1; SMN2MAPT
SCHEMBL21551921 0.79 HDAC1 (0.57) CYP1A2ALDH1A1HPGDLMNASETD7
SCHEMBL21551983 0.78 CYP1A2 (0.54) CYP1A2ALDH1A1HPGDKDM4EGLA
SCHEMBL21568019 0.78 ALDH1A1 (0.56) CYP1A2ALDH1A1HPGDKDM4ELMNA
SCHEMBL22708463 0.77 ALDH1A1 (0.57) ALDH1A1HPGDKDM4ELMNAGLA
SCHEMBL21552087 0.75 MCHR1 (0.54) ALDH1A1HPGDSETD7ALOX5TMEM97
SCHEMBL6642558 0.75 ALDH1A1 (0.55) ALDH1A1HPGDKDM4ESETD7SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019216810-A1 NEW ANTIFUNGAL COMPOUNDS URBAN CONSTANTIN (SE) 2019-11-14 WO claimed
WO-2019216810-A1 NEW ANTIFUNGAL COMPOUNDS URBAN CONSTANTIN (SE) 2019-11-14 WO disclosed
WO-2019216810-A1 NEW ANTIFUNGAL COMPOUNDS URBAN CONSTANTIN (SE) 2019-11-14 WO disclosed