SCHEMBL21551941

SCHEMBL21551941

CN1CCN(CCNC(=O)c2ccc(/C=C/c3ccc(Br)cc3Br)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.62
HDAC2 Q92769 1/20 0.62
HDAC8 Q9BY41 1/20 0.62
RAD52 P43351 1/20 0.48
ABL1 P00519 1/20 0.47
BCR P11274 1/20 0.47
MAPT P10636 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
NAMPT P43490 1/20 0.44
TSHR P16473 1/20 0.44
IKBKE Q14164 1/20 0.44
TBK1 Q9UHD2 1/20 0.44
PLD2 O14939 2/20 0.43
PLD1 Q13393 2/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
HTR1B P28222 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21551983 0.91 CYP1A2 (0.54) HDAC6HDAC2HDAC8MAPTNPSR1
SCHEMBL21551975 0.89 TSHR (0.59) HDAC6HDAC2HDAC8ABL1TSHR
SCHEMBL21551964 0.84 TSHR (0.54) MAPTNAMPTTSHRDRD2DRD3
SCHEMBL21551954 0.83 TSHR (0.69) MAPTTSHR
SCHEMBL21551957 0.80 HDAC2 (0.59) HDAC6HDAC2HDAC8RAD52MAPT
SCHEMBL21551953 0.79 CYP1A2 (0.50) MAPT
SCHEMBL21551981 0.76 LMNA (0.52) HDAC6HDAC2HDAC8RAD52MAPT
SCHEMBL21568402 0.74 ALDH1A1 (0.52) HDAC6HDAC2HDAC8RAD52MAPT
SCHEMBL11983548 0.73 HDAC2 (0.78) HDAC6HDAC2HDAC8RAD52NPSR1
SCHEMBL21568404 0.72 ALDH1A1 (0.49) HDAC6HDAC2HDAC8PLD2PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019216810-A1 NEW ANTIFUNGAL COMPOUNDS URBAN CONSTANTIN (SE) 2019-11-14 WO claimed
WO-2019216810-A1 NEW ANTIFUNGAL COMPOUNDS URBAN CONSTANTIN (SE) 2019-11-14 WO disclosed