SCHEMBL21554572

SCHEMBL21554572

COc1cc(CN(C)CC2CC2)cc(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPK1 P28482 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CALM1 P0DP23 1/20 0.40
KDR P35968 1/20 0.39
FLT3 P36888 1/20 0.39
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
TACR1 P25103 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23507263 0.76 TSHR (0.56) TSHRALDH1A1MAPK1KDM4ECALM1
SCHEMBL21554823 0.75 ALDH1A1 (0.41) TSHRALDH1A1KDM4EHSD17B10CALM1
SCHEMBL3100529 0.73 ALDH1A1 (0.52) TSHRALDH1A1MAPK1CALM1GAA
SCHEMBL23507393 0.73 GRIN2D (0.51) TSHRALDH1A1MAPK1CALM1GRIN2D
SCHEMBL14045705 0.71 ALDH1A1 (0.52) TSHRALDH1A1KDM4E
SCHEMBL16327151 0.69 PYCR1 (0.50)
SCHEMBL15746871 0.69 TSHR (0.47) TSHRALDH1A1MAPK1HSD17B10CALM1
SCHEMBL17887960 0.68 PYCR1 (0.51) MEN1KMT2A
SCHEMBL4267535 0.68 CXCR3 (0.41) TSHRALDH1A1
SCHEMBL1240985 0.68 PYCR1 (0.51) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2776408-B1 ANTICANCER BENZOPYRAZINES VIA THE INHIBITION OF FGFR KINASES ASTEX THERAPEUTICS LTD (GB) 2019-11-06 EP disclosed