SCHEMBL21574568

SCHEMBL21574568

Cc1ccc2nc(Cl)c(Cc3ccc(C(F)(F)F)s3)c(Cl)c2c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.40
ELANE P08246 1/20 0.39
RORC P51449 7/20 0.38
RXFP1 Q9HBX9 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 3/20 0.36
MAPT P10636 3/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.34
HTT P42858 1/20 0.34
NCOA1 Q15788 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34
ADRB2 P07550 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16633163 0.86 RORC (0.38) RORCRXFP1CYP1A2CYP2D6CYP2C9
SCHEMBL16662148 0.76 RORC (0.56) PKMELANERORCRXFP1CYP1A2
SCHEMBL16632876 0.75 RORC (0.44) RORC
SCHEMBL16632926 0.72 ALDH1A1 (0.44) RORCCYP1A2CYP2C9CYP2C19LMNA
SCHEMBL5085893 0.67 LMNA (0.54) PKMELANELMNAMAPTKDM4E
SCHEMBL14044130 0.67 CYP1A2 (0.72) PKMELANERXFP1CYP1A2CYP2D6
SCHEMBL16632741 0.65 RORC (0.42) PKMRORCRXFP1CYP1A2CYP2D6
SCHEMBL9593290 0.65 LMNA (0.62) PKMELANECYP1A2LMNAMAPT
SCHEMBL16656034 0.64 RORC (0.67) RORC
SCHEMBL27138975 0.64 LMNA (0.49) ELANELMNAMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057951-B1 METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T JANSSEN PHARMACEUTICA NV (BE) 2019-11-20 EP disclosed